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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $34.85 | Total: $174.25 |
| 1 | 10 | $29.52 | Total: $295.20 |
| 1 | 25 | $25.01 | Total: $625.25 |
| 1 | 50 | $21.32 | Total: $1,066.00 |
| 1 | 100 | $18.45 | Total: $1,845.00 |
Overview
BL-1249 is a selective and potent non-steroidal potassium channel activator with anti-inflammatory activity that activates K2P2.1 (TREK-1) and K2P10.1 (TREK-2).
Chemical Properties
| Molecular Formula | C17H17N5 |
| Molecular Weight | 291.35 |
| CAS Numbers | 18200-13-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C1CCc2c(C1)cccc2Nc1ccccc1-c1nnn[nH]1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Pope L, et al. Protein and Chemical Determinants of BL-1249 Action and Selectivity for K2P Channels. ACS Chem Neurosci. 2018 Dec 19;9[12] 3153-3165.