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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $39.95 | Total: $199.75 |
| 1 | 10 | $33.84 | Total: $338.40 |
| 1 | 25 | $28.67 | Total: $716.75 |
| 1 | 50 | $24.44 | Total: $1,222.00 |
| 1 | 100 | $21.15 | Total: $2,115.00 |
Overview
P-1075 is a potent sulfonylurea receptor 2-associated ATP-sensitive potassium channels (SUR2-KIR6) activator (EC50 = 45 nM). P-1075 opens opens mitoKATP channels and may be cardioprotective.
Chemical Properties
| Molecular Formula | C12H17N5 |
| Molecular Weight | 231.3 |
| CAS Numbers | 60559-98-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCC(C)(C)NC(NC#N)=Nc1cccnc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Schwanstecher M, et al. Potassium channel openers require ATP to bind to and act through sulfonylurea receptors. EMBO J. 1998 Oct 1;17[19] 5529-35.