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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $144.50 | Total: $722.50 |
| 1 | 10 | $122.40 | Total: $1,224.00 |
| 1 | 25 | $103.70 | Total: $2,592.50 |
| 1 | 50 | $88.40 | Total: $4,420.00 |
| 1 | 100 | $76.50 | Total: $7,650.00 |
Overview
CHET3 is a highly selective allosteric activator for TASK-3-containing K2P channels. CHET3 has shown potent in vivo analgesic effects in various acute and chronic pain models in rodents.
Chemical Properties
| Molecular Formula | C21H21N5O3S |
| Molecular Weight | 423.49 |
| CAS Numbers | 2489231-47-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(C(NC=1NC(CSC2=CC=C(C)C=C2)=CC(=O)N1)=N)C=3C=C4C(=CC3)OCCO4 |
Storage and Handling
0C Short Term, -20C Long Term
References
Liao P, et al. Selective activation of TWIK-related acid-sensitive K+ 3 subunit-containing channels is analgesic in rodent models. Sci Transl Med. 2019 Nov 20;11[519] eaaw8434.