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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $69.70 | Total: $348.50 |
| 1 | 10 | $59.04 | Total: $590.40 |
| 1 | 25 | $50.02 | Total: $1,250.50 |
| 1 | 50 | $42.64 | Total: $2,132.00 |
| 1 | 100 | $36.90 | Total: $3,690.00 |
Overview
TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the intermediate (IM) state of TREK-1.
Chemical Properties
| Molecular Formula | C18H14ClN3O2S |
| Molecular Weight | 371.84 |
| CAS Numbers | 326921-25-9 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | S(CC(NNC(=O)C1=CC=C(Cl)C=C1)=O)C2=NC3=C(C=C2)C=CC=C3 |
Storage and Handling
0C Short Term, -20C Long Term
References
Ma Y , Luo Q , Fu J , et al. Discovery of an Inhibitor for the TREK-1 Channel Targeting an Intermediate Transition State of Channel Gating[J]. Journal of Medicinal Chemistry, 2020.