CVT-313

CVT-313

AOB1132

CAS: 199986-75-9

 

Chemical Name: 2-[2-Hydroxyethyl-[6-[(4-methoxyphenyl)methylamino]-9-propan-2-ylpurin-2-yl]amino]ethanol

More details

1000 Items

$27.30

$27.30 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $17.85 Total: $89.25
110 $15.12 Total: $151.20
125 $12.81 Total: $320.25
150 $10.92 Total: $546.00
1100 $9.45 Total: $945.00

Overview

Specific inhibitor of CDK2/cyclin A and CDK2/cyclin E

Chemical Properties

Molecular FormulaC20H28N6O3
Molecular Weight400.5
CAS Numbers199986-75-9
SolubilityDMSO
Purity95% by HPLC
IUPAC/Chemical Name2,2'-[[6-[[(4-methoxyphenyl)methyl]amino]-9-(1-methylethyl)-9H-purin-2-yl]imino]bis-ethanol
InChl KeyNQVIIUBWMBHLOZ-UHFFFAOYSA-N
InChl CodeInChI=1S/C20H28N6O3/c1-14(2)26-13-22-17-18(21-12-15-4-6-16(29-3)7-5-15)23-20(24-19(17)26)25(8-10-27)9-11-28/h4-7,13-14,27-28H,8-12H2,1-3H3,(H,21,23,24)
SMILES CodeOCCN(CCO)C1=NC(N(C(C)C)C=N2)=C2C(NCC3=CC=C(OC)C=C3)=N1

Storage and Handling

0°C (short term), -20°C (long term), desiccated

Synonyms

CVT 313; CVT313

References

1) Brooks, E.E., Gray, N.S., Joly, A.H., et al. CVT-313, a specific and potent inhibitor of CDK2 that prevents neointimal proliferation. J. Biol. Chem. 272(46), 29207-29211 (1997).

2) Bhattacharjee, R.N., Banks, G.C., Trotter, K.W., et al. Histone H1 phosphorylation by Cdk2 selectively modulates mouse mammary tumor virus transcription through chromatin remodeling. Mol. Cell. Biol. 21(16), 5417-5454 (2001).