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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $27.20 | Total: $136.00 |
| 1 | 10 | $23.04 | Total: $230.40 |
| 1 | 25 | $19.52 | Total: $488.00 |
| 1 | 50 | $16.64 | Total: $832.00 |
| 1 | 100 | $14.40 | Total: $1,440.00 |
Overview
(EZ)-Zotiraciclib ((EZ)-TG02) effectively inhibits CDK2, JAK2, and FLT3 with IC50s of 13 nM, 73 nM, and 56 nM, respectively.
Chemical Properties
| Molecular Formula | C23H24N4O |
| Molecular Weight | 372.46 |
| CAS Numbers | 937270-47-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN1CC2=CC(N=C3NC(C=4C=C(C=CC4)OCCC=CC1)=CC=N3)=CC=C2 |
Storage and Handling
0C Short Term, -20C Long Term
References
William AD, et al. Discovery of kinase spectrum selective macrocycle [16E]-14-methyl-20-oxa-5,7,14,26-tetraazatetracyclo[19.3.1.1[2,6].1[8,12]]heptacosa-1[25],2[26],3,5,8[27],9,11,16,21,23-decaene [SB1317TG02], a potent inhibitor of cyclin dependent kina