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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $106.25 | Total: $531.25 |
| 1 | 10 | $90.00 | Total: $900.00 |
| 1 | 25 | $76.25 | Total: $1,906.25 |
| 1 | 50 | $65.00 | Total: $3,250.00 |
| 1 | 100 | $56.25 | Total: $5,625.00 |
Overview
GSK-3? inhibitor 14 (1,5-Benzothiazepin-4(5H)-one, 2,3-dihydro-2-methyl-5-(phenylmethyl)-) is a weak GSK-3? inhibitor, IC50? 100?M.
Chemical Properties
| Molecular Formula | C17H17NOS |
| Molecular Weight | 283.39 |
| CAS Numbers | 863004-48-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(N1C=2C(SC(C)CC1=O)=CC=CC2)C3=CC=CC=C3 |
Storage and Handling
0C Short Term, -20C Long Term
References
Zhang P, et al. Design, synthesis and biological evaluation of benzothiazepinones [BTZs] as novel non-ATP competitive inhibitors of glycogen synthase kinase-3? [GSK-3?]. Eur J Med Chem. 2013 Mar;61 95-103.