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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $136.00 | Total: $680.00 |
| 1 | 10 | $115.20 | Total: $1,152.00 |
| 1 | 25 | $97.60 | Total: $2,440.00 |
| 1 | 50 | $83.20 | Total: $4,160.00 |
| 1 | 100 | $72.00 | Total: $7,200.00 |
Overview
IKK2-IN-4(IKK2 Inhibitor VI) is a highly potent IKK-2 inhibitor with an IC50 value of 25 nM. IKK2-IN-4 inhibited the production of TNF-? in PBMC induced by LPS.
Chemical Properties
| Molecular Formula | C12H11N3O2S |
| Molecular Weight | 261.3 |
| CAS Numbers | 354811-10-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(C(N)=O)C=1SC(=CC1C(N)=O)C2=CC=CC=C2 |
Storage and Handling
0C Short Term, -20C Long Term
References
Baxter A, et, al. Hit-to-lead studies the discovery of potent, orally active, thiophenecarboxamide IKK-2 inhibitors. Bioorg Med Chem Lett. 2004 Jun 7;14[11] 2817-22.