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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $27.20 | Total: $136.00 |
| 1 | 10 | $23.04 | Total: $230.40 |
| 1 | 25 | $19.52 | Total: $488.00 |
| 1 | 50 | $16.64 | Total: $832.00 |
| 1 | 100 | $14.40 | Total: $1,440.00 |
Overview
Tanzisertib (CC-930) (CC-930) is a potent inhibitor of JNK123 with IC50s of 6176 nM, respectively, with potential antifibrotic activity.
Chemical Properties
| Molecular Formula | C21H23F3N6O2 |
| Molecular Weight | 448.44 |
| CAS Numbers | 899805-25-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.OC1CCC(CC1)Nc1ncc2nc(Nc3c(F)cc(F)cc3F)n([C@H]3CCOC3)c2n1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Plantevin Krenitsky V, et al. Discovery of CC-930, an orally active anti-fibrotic JNK inhibitor. Bioorg Med Chem Lett. 2012 Feb 1;22[3] 1433-8.