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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.10 | Total: $110.50 |
| 1 | 10 | $18.72 | Total: $187.20 |
| 1 | 25 | $15.86 | Total: $396.50 |
| 1 | 50 | $13.52 | Total: $676.00 |
| 1 | 100 | $11.70 | Total: $1,170.00 |
Overview
Trilaciclib hydrochloride (G1T28 hydrochloride) is an inhibitor of CDK46 (IC50s: 1 nM and 4 nM for CDK4 and CDK6).
Chemical Properties
| Molecular Formula | C24H32Cl2N8O |
| Molecular Weight | 519.47 |
| CAS Numbers | 1977495-97-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.Cl.CN1CCN(CC1)c1ccc(Nc2ncc3cc4C(=O)NCC5(CCCCC5)n4c3n2)nc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Bisi JE, et al. Preclinical Characterization of G1T28 A Novel CDK46 Inhibitor for Reduction of Chemotherapy-Induced Myelosuppression. Mol Cancer Ther. 2016 May;15[5] 783-93.