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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $116.45 | Total: $582.25 |
| 1 | 10 | $98.64 | Total: $986.40 |
| 1 | 25 | $83.57 | Total: $2,089.25 |
| 1 | 50 | $71.24 | Total: $3,562.00 |
| 1 | 100 | $61.65 | Total: $6,165.00 |
Overview
GKI-1 HCl is a Greatwall (GWL) kinase inhibitor that inhibits hGWLFL and hGWL-KinDom.The inhibitory effect of GKI-1 HCl on ROCK1 is more significant.
Chemical Properties
| Molecular Formula | C15H13Cl2N3 |
| Molecular Weight | 306.19 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | ClC1=CC=C(NC2=CC=CC(C3=CNN=C3)=C2)C=C1.Cl |
Storage and Handling
0C Short Term, -20C Long Term
References
Ocasio CA, et al. A first generation inhibitor of human Greatwall kinase, enabled by structural and functional characterisation of a minimal kinase domain construct. Oncotarget. 2016;7[44] 71182-71197.