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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.95 | Total: $114.75 |
| 1 | 10 | $19.44 | Total: $194.40 |
| 1 | 25 | $16.47 | Total: $411.75 |
| 1 | 50 | $14.04 | Total: $702.00 |
| 1 | 100 | $12.15 | Total: $1,215.00 |
Overview
GW843682X (GW843682) is a selective and ATP-competitive inhibitor of PLK1 and PLK3 (IC50s = 2.2 nM and 9.1 nM).
Chemical Properties
| Molecular Formula | C22H18F3N3O4S |
| Molecular Weight | 477.46 |
| CAS Numbers | 660868-91-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1cc2ncn(-c3cc(OCc4ccccc4C(F)(F)F)c(s3)C(N)=O)c2cc1OC |
Storage and Handling
0C Short Term, -20C Long Term
References
Didier C, et al. Evaluation of Polo-like Kinase 1 inhibition on the G2M checkpoint in Acute Myelocytic Leukaemia. Eur J Pharmacol. 2008 Sep 4;591[1-3] 102-5.