Categories
- PROTAC Linker
- Protein Control Ligand
- Pathway Inhibitors
- Function Modulators
- Activators
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- Nuclear Receptor Ligands
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $107.10 | Total: $535.50 |
| 1 | 10 | $90.72 | Total: $907.20 |
| 1 | 25 | $76.86 | Total: $1,921.50 |
| 1 | 50 | $65.52 | Total: $3,276.00 |
| 1 | 100 | $56.70 | Total: $5,670.00 |
Overview
Parsaclisib (INCB050465) is a potent and selective inhibitor of PI3K?(IC50 of 1 nM at 1 mM ATP)
Chemical Properties
| Molecular Formula | C20H22ClFN6O2 |
| Molecular Weight | 432.88 |
| CAS Numbers | 1426698-88-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCOc1c(cc(Cl)c(F)c1[C@@H]1CNC(=O)C1)[C@H](C)n1nc(C)c2c(N)ncnc12 |
Storage and Handling
0C Short Term, -20C Long Term
References
Niu Shin, et al. Abstract 2671 INCB050465, a novel PI3K? inhibitor, synergizes with PIM protein kinase inhibition to cause tumor regression in a model of DLBCL. Cancer Research. 2015, Aug. 75[15].