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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $64.60 | Total: $323.00 |
| 1 | 10 | $54.72 | Total: $547.20 |
| 1 | 25 | $46.36 | Total: $1,159.00 |
| 1 | 50 | $39.52 | Total: $1,976.00 |
| 1 | 100 | $34.20 | Total: $3,420.00 |
Overview
JNK-IN-7 (JNK inhibitor) is a selective JNK123 inhibitor (IC50: 1.541.990.75 nM). It can also inhibit phosphorylation of c-Jun, which is a substrate of JNK kinase.
Chemical Properties
| Molecular Formula | C28H27N7O2 |
| Molecular Weight | 493.56 |
| CAS Numbers | 1408064-71-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN(C)CC=CC(=O)Nc1cccc(c1)C(=O)Nc1ccc(Nc2nccc(n2)-c2cccnc2)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Zhang T, et al. Discovery of Potent and Selective Covalent Inhibitors of JNK. Chem Biol. 2012 Jan 27;19[1] 140-54.