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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $61.20 | Total: $306.00 |
| 1 | 10 | $51.84 | Total: $518.40 |
| 1 | 25 | $43.92 | Total: $1,098.00 |
| 1 | 50 | $37.44 | Total: $1,872.00 |
| 1 | 100 | $32.40 | Total: $3,240.00 |
Overview
Refametinib R enantiomer (RDEA119 R enantiomer) is an MEK inhibitor with an EC50 of 2.0-15 nM.Refametinib (R enantiomer) has anticancer activity and can be used in cancer research.
Chemical Properties
| Molecular Formula | C19H20F3IN2O5S |
| Molecular Weight | 572.34 |
| CAS Numbers | 923032-38-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | S(NC1=C(NC2=C(F)C=C(I)C=C2)C(F)=C(F)C=C1OC)(=O)(=O)C3(C[C@H](CO)O)CC3 |
Storage and Handling
0C Short Term, -20C Long Term
References
Andreas Maderna, et al. N-[arylamino]-sulfonamide inhibitors of mek. WO 2007014011 A2.