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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $495.55 | Total: $2,477.75 |
| 1 | 10 | $419.76 | Total: $4,197.60 |
| 1 | 25 | $355.63 | Total: $8,890.75 |
| 1 | 50 | $303.16 | Total: $15,158.00 |
| 1 | 100 | $262.35 | Total: $26,235.01 |
Overview
AY 77 (Unk-Cha-Chg-NH2) is a potent and selective PAR2 agonist. AY 77 showed selectivity for Ca2+ and ERK12 signaling (ec50 value of Ca2+ release was 40 nM and ec50 value of ERK12 phosphorylation was 2 ?M). AY 77 can promote migration of human breast cancer cells in vitro.
Chemical Properties
| Molecular Formula | C21H32N4O4 |
| Molecular Weight | 404.5 |
| CAS Numbers | 1835734-92-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | [C@H](CC1CCCCC1)(C(N[C@H](C(N)=O)[C@@H]2CCCCC2)=O)NC(=O)C3=CC=NO3 |
Storage and Handling
0C Short Term, -20C Long Term
References
Jiang Y, et al. Biased Signaling by Agonists of Protease Activated Receptor 2. ACS Chem Biol. 2017;12[5] 1217-1226.