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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $126.65 | Total: $633.25 |
| 1 | 10 | $107.28 | Total: $1,072.80 |
| 1 | 25 | $90.89 | Total: $2,272.25 |
| 1 | 50 | $77.48 | Total: $3,874.00 |
| 1 | 100 | $67.05 | Total: $6,705.00 |
Overview
BAY-985 is a potent, selective, and orally active ATP-competitive dual inhibitor of TBK1 and IKK? (IC50s: 230 and 2 nM for TBK1 (lowhigh ATP) and IKK?) with antitumor efficacy.
Chemical Properties
| Molecular Formula | C27H30F3N9O |
| Molecular Weight | 553.58 |
| CAS Numbers | 2409479-29-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C[C@@H](N1CCN(CC1)C(=O)CC(F)(F)F)c1ccnc(Nc2nc3ccc(cc3[nH]2)-c2cc(ncn2)N(C)C)c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Lefranc J, et al. Discovery of BAY-985, a Highly Selective TBK1IKK? Inhibitor. J Med Chem. 2020 Jan 10.