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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $64.60 | Total: $323.00 |
| 1 | 10 | $54.72 | Total: $547.20 |
| 1 | 25 | $46.36 | Total: $1,159.00 |
| 1 | 50 | $39.52 | Total: $1,976.00 |
| 1 | 100 | $34.20 | Total: $3,420.00 |
Overview
CDK8-IN-1 is a selective CDK8 inhibitor (IC50: 3 nM).
Chemical Properties
| Molecular Formula | C11H8F3N3O |
| Molecular Weight | 255.2 |
| CAS Numbers | 1629633-48-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | NC(=O)c1[nH]cc(c1C(F)(F)F)-c1ccncc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Han X, et al. Discovery of potent and selective CDK8 inhibitors through FBDD approach. Bioorg Med Chem Lett. 2017 Sep 15;27[18] 4488-4492.