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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $141.10 | Total: $705.50 |
| 1 | 10 | $119.52 | Total: $1,195.20 |
| 1 | 25 | $101.26 | Total: $2,531.50 |
| 1 | 50 | $86.32 | Total: $4,316.00 |
| 1 | 100 | $74.70 | Total: $7,470.00 |
Overview
CHK1-IN-3 is an inhibitor of checkpoint kinase 1 (CHK1; IC50: 0.4 nM).
Chemical Properties
| Molecular Formula | C20H23N9O |
| Molecular Weight | 405.46 |
| CAS Numbers | 2097252-39-4 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N(C)C=1C(=CN=C(NC=2C=C(O[C@@H]3CCCNC3)C(C#N)=NC2)N1)C4=CN(C)N=C4 |
Storage and Handling
0C Short Term, -20C Long Term
References
Tong L, et al. Discovery of [R]-5-[[5-[1-methyl-1H-pyrazol-4-yl]-4-[methylamino]pyrimidin-2-yl]amino]-3-[piperidin-3-yloxy]picolinonitrile, a novel CHK1 inhibitor for hematologic malignancies. Eur J Med Chem. 2019 Jul 1;173 44-62.