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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $34.85 | Total: $174.25 |
| 1 | 10 | $29.52 | Total: $295.20 |
| 1 | 25 | $25.01 | Total: $625.25 |
| 1 | 50 | $21.32 | Total: $1,066.00 |
| 1 | 100 | $18.45 | Total: $1,845.00 |
Overview
G-5555 is a potent inhibitor of p21-activated kinase 1 (PAK1) (Kis: 3.7 nM and 11 nM for PAK1 and PAK2, respectively).
Chemical Properties
| Molecular Formula | C25H25ClN6O3 |
| Molecular Weight | 492.96 |
| CAS Numbers | 1648863-90-4 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CNc1ncc2cc(-c3ccc(cc3Cl)-c3cccc(C)n3)c(=O)n(C[C@H]3OC[C@H](N)CO3)c2n1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Ndubaku CO, et al. Design of Selective PAK1 Inhibitor G-5555 Improving Properties by Employing an Unorthodox Low-pK a Polar Moiety. ACS Med Chem Lett. 2015 Oct 31;6[12] 1241-6.