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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $153.85 | Total: $769.25 |
| 1 | 10 | $130.32 | Total: $1,303.20 |
| 1 | 25 | $110.41 | Total: $2,760.25 |
| 1 | 50 | $94.12 | Total: $4,706.00 |
| 1 | 100 | $81.45 | Total: $8,145.00 |
Overview
LDH-IN-1 is a pyrazole-based human lactate dehydrogenase (LDH) inhibitor(IC50s of 32 and 27 nM for LDHA and LDHB, respectively).
Chemical Properties
| Molecular Formula | C30H26N4O4S2 |
| Molecular Weight | 570.68 |
| CAS Numbers | 1964515-43-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | NS(=O)(=O)c1ccc(Cc2c(CC3CC3)n(nc2-c2cccc(c2)-c2ccccc2)-c2nc(cs2)C(O)=O)cc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Rai G, et al. Discovery and Optimization of Potent, Cell-Active Pyrazole-Based Inhibitors of Lactate Dehydrogenase [LDH]. J Med Chem. 2017 Nov 22;60[22] 9184-9204.