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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $85.85 | Total: $429.25 |
| 1 | 10 | $72.72 | Total: $727.20 |
| 1 | 25 | $61.61 | Total: $1,540.25 |
| 1 | 50 | $52.52 | Total: $2,626.00 |
| 1 | 100 | $45.45 | Total: $4,545.00 |
Overview
ROCK-IN-1, a potent ROCK inhibitor, effectively inhibits ROCK2-mediated signaling with an IC50 value of 1.2 nM. ROCK-IN-1 is applicable in the study of neurological disorders and inflammation-related diseases.
Chemical Properties
| Molecular Formula | C20H18FN3O |
| Molecular Weight | 335.37 |
| CAS Numbers | 934387-35-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(N)c1ccc(cc1-c1ccc(F)cc1)C(=O)Nc1ccncc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Boland S, et al. 3-[2-[Aminomethyl]-5-[[pyridin-4-yl]carbamoyl]phenyl] benzoates as soft ROCK inhibitors. Bioorg Med Chem Lett. 2013 Dec 1;23[23] 6442-6.