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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $48.45 | Total: $242.25 |
| 1 | 10 | $41.04 | Total: $410.40 |
| 1 | 25 | $34.77 | Total: $869.25 |
| 1 | 50 | $29.64 | Total: $1,482.00 |
| 1 | 100 | $25.65 | Total: $2,565.00 |
Overview
AZD 4017 is an inhibitor of 11?-Hydroxysteroid Dehydrogenase Type 1(11?-HSD1) (IC50: 7 nM).
Chemical Properties
| Molecular Formula | C22H33N3O3S |
| Molecular Weight | 419.58 |
| CAS Numbers | 1024033-43-9 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CCCSc1nc(ccc1C(=O)NC1CCCCC1)N1CCC[C@@H](CC(O)=O)C1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Scott JS, et al. Discovery of a potent, selective, and orally bioavailable acidic 11?-hydroxysteroid dehydrogenase type 1 [11?-HSD1] inhibitor discovery of 2-[[3S]-1-[5-[cyclohexylcarbamoyl]-6-propylsulfanylpyridin-2-yl]-3-piperidyl]acetic acid [AZD4017]. J Med Chem. 2012 Jun 28;55[12] 5951-64.