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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $26.35 | Total: $131.75 |
| 1 | 10 | $22.32 | Total: $223.20 |
| 1 | 25 | $18.91 | Total: $472.75 |
| 1 | 50 | $16.12 | Total: $806.00 |
| 1 | 100 | $13.95 | Total: $1,395.00 |
Overview
BMS-935177 is a reversible BTK inhibitor with IC50 value of 3 nM.
Chemical Properties
| Molecular Formula | C31H26N4O3 |
| Molecular Weight | 502.56 |
| CAS Numbers | 1231889-53-4 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1c(cccc1-n1cnc2ccccc2c1=O)-c1ccc(C(N)=O)c2[nH]c3cc(ccc3c12)C(C)(C)O |
Storage and Handling
0C Short Term, -20C Long Term
References
De Lucca GV, et al. Small Molecule Reversible Inhibitors of Bruton's Tyrosine Kinase [BTK] Structure-Activity Relationships Leading to the Identification of 7-[2-Hydroxypropan-2-yl]-4-[2-methyl-3-[4-oxo-3,4-dihydroquinazolin-3-yl]phenyl]-9H-carbazole-1-carboxamide [BMS-935177]. J Med Chem. 2016 Sep 8;59[17] 7915-35.