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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.10 | Total: $110.50 |
| 1 | 10 | $18.72 | Total: $187.20 |
| 1 | 25 | $15.86 | Total: $396.50 |
| 1 | 50 | $13.52 | Total: $676.00 |
| 1 | 100 | $11.70 | Total: $1,170.00 |
Overview
CGP60474 is an inhibitor of VEGFR-2 (IC50 = 84 nM) and an inhibitor of ATP-competitive PKC. CGP60474 is also a highly potent anti-endotoxemic agent and inhibits cyclin-dependent kinase (CDK) potently.
Chemical Properties
| Molecular Formula | C18H18ClN5O |
| Molecular Weight | 355.82 |
| CAS Numbers | 164658-13-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | OCCCNc1cc(ccn1)-c1ccnc(Nc2cccc(Cl)c2)n1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Kuo GH, et al. Synthesis and identification of [1,3,5]triazine-pyridine biheteroaryl as a novel series of potent cyclin-dependent kinase inhibitors. J Med Chem. 2005 Jul 14;48[14] 4535-46.