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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $69.70 | Total: $348.50 |
| 1 | 10 | $59.04 | Total: $590.40 |
| 1 | 25 | $50.02 | Total: $1,250.50 |
| 1 | 50 | $42.64 | Total: $2,132.00 |
| 1 | 100 | $36.90 | Total: $3,690.00 |
Overview
YKL-5-124, a potent, selective and covalent CDK7 inhibitor with an IC50 of 9.7 nM, 1300 nM and 3020 nM for CDK7Mat1CycH, CDK2 and CDK9 respectively, displays biochemical and cellular selectivity for CDK7 over CDK1213.
Chemical Properties
| Molecular Formula | C28H33N7O3 |
| Molecular Weight | 515.61 |
| CAS Numbers | 1957203-01-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN(C)C[C@@H](NC(=O)N1Cc2c(NC(=O)c3ccc(NC(=O)C=C)cc3)n[nH]c2C1(C)C)c1ccccc1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Olson CM, Liang Y, Leggett A, Park WD, Li L, Mills CE, Elsarrag SZ, Ficarro SB, Zhang T, D