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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $27.20 | Total: $136.00 |
| 1 | 10 | $23.04 | Total: $230.40 |
| 1 | 25 | $19.52 | Total: $488.00 |
| 1 | 50 | $16.64 | Total: $832.00 |
| 1 | 100 | $14.40 | Total: $1,440.00 |
Overview
SM 16 is an ALK5ALK4 kinase inhibitor with Ki values of 10 nM and 1.5 nM, respectively.
Chemical Properties
| Molecular Formula | C25H26N4O3 |
| Molecular Weight | 430.5 |
| CAS Numbers | 614749-78-9 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cc1cccc(n1)-c1[nH]c(nc1-c1ccc2OCOc2c1)C12CCC(CC1)(CC2)C(N)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Suzuki E, et al. A novel small-molecule inhibitor of transforming growth factor beta type I receptor kinase [SM16] inhibits murine mesothelioma tumor growth in vivo and prevents tumor recurrence after surgical resection. Cancer Res. 2007 Mar 1;67[5] 2351-9.