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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $34.85 | Total: $174.25 |
| 1 | 10 | $29.52 | Total: $295.20 |
| 1 | 25 | $25.01 | Total: $625.25 |
| 1 | 50 | $21.32 | Total: $1,066.00 |
| 1 | 100 | $18.45 | Total: $1,845.00 |
Overview
ERK5-IN-1 is a potent ERK5 inhibitor (IC50: 87 nM) and also inhibits LRRK2[G2019S] (IC50: 26 nM).
Chemical Properties
| Molecular Formula | C25H29N7O2 |
| Molecular Weight | 459.54 |
| CAS Numbers | 1234479-76-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1cc(ccc1Nc1ncc2N(C)C(=O)c3ccccc3N(C)c2n1)N1CCN(C)CC1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Deng X, et al. Structural determinants for ERK5 [MAPK7] and leucine rich repeat kinase 2 activities of benzo[e]pyrimido-[5,4-b]diazepine-6[11H]-ones. Eur J Med Chem. 2013;70 758-767.