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- Protein Control Ligand
- Pathway Inhibitors
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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.10 | Total: $110.50 |
| 1 | 10 | $18.72 | Total: $187.20 |
| 1 | 25 | $15.86 | Total: $396.50 |
| 1 | 50 | $13.52 | Total: $676.00 |
| 1 | 100 | $11.70 | Total: $1,170.00 |
Overview
Longdaysin is an inhibitor of CK1? and CK1? (IC50s: 5.68.8 ?M). It also can inhibit ERK2 (IC50: 52 ?M).
Chemical Properties
| Molecular Formula | C16H16F3N5 |
| Molecular Weight | 335.33 |
| CAS Numbers | 1353867-91-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(C)n1cnc2c(NCc3cccc(c3)C(F)(F)F)ncnc12 |
Storage and Handling
0C Short Term, -20C Long Term
References
Hirota T, et al. High-throughput chemical screen identifies a novel potent modulator of cellular circadian rhythms and reveals CKI? as a clock regulatory kinase. PLoS Biol. 2010 Dec 14;8[12] e1000559.