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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $36.55 | Total: $182.75 |
| 1 | 10 | $30.96 | Total: $309.60 |
| 1 | 25 | $26.23 | Total: $655.75 |
| 1 | 50 | $22.36 | Total: $1,118.00 |
| 1 | 100 | $19.35 | Total: $1,935.00 |
Overview
Senexin A is an effective and selective CDK8 inhibitor that also inhibits CDK19 with Kd values of 0.83 microns and 0.31 microns, respectively.
Chemical Properties
| Molecular Formula | C17H14N4 |
| Molecular Weight | 274.32 |
| CAS Numbers | 1366002-50-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | N#Cc1ccc2ncnc(NCCc3ccccc3)c2c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Porter D C , Farmaki E , Altilia S , et al. Cyclin-dependent kinase 8 mediates chemotherapy-induced tumor-promoting paracrine activities[J]. Proceedings of the National Academy of Sciences, 2012, 109[34] 13799-13804.