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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $23.80 | Total: $119.00 |
| 1 | 10 | $20.16 | Total: $201.60 |
| 1 | 25 | $17.08 | Total: $427.00 |
| 1 | 50 | $14.56 | Total: $728.00 |
| 1 | 100 | $12.60 | Total: $1,260.00 |
Overview
PI3KAktmTOR-IN-2 is a potent PI3KAKTmTOR inhibitor with anticancer effects and selectivity for MDA-MB-231 cells (IC50 2.29 ?M). It induces cell cycle arrest and apoptosis in cancer cells.
Chemical Properties
| Molecular Formula | C17H13F2NO |
| Molecular Weight | 285.29 |
| CAS Numbers | 2757804-89-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Fc1cc(F)cc(c1)C1OCCc2c1[nH]c1ccccc21 |
Storage and Handling
0C Short Term, -20C Long Term
References
Qin J, et al. Design, synthesis and biological evaluation of novel 1,3,4,9-tetrahydropyrano[3,4-b]indoles as potential treatment of triple negative breast cancer by suppressing PI3KAKTmTOR pathway. Bioorg Med Chem. 2021 Dec 31;55 116594.