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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $56.10 | Total: $280.50 |
| 1 | 10 | $47.52 | Total: $475.20 |
| 1 | 25 | $40.26 | Total: $1,006.50 |
| 1 | 50 | $34.32 | Total: $1,716.00 |
| 1 | 100 | $29.70 | Total: $2,970.00 |
Overview
A-674563 2HCl is an Akt1 inhibitor with Ki of 11 nM, modest potent to PKA and >30-fold selective for Akt1 over PKC.
Chemical Properties
| Molecular Formula | C22H24Cl2N4O |
| Molecular Weight | 431.36 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.Cl.Cc1n[nH]c2ccc(cc12)-c1cncc(OC[C@@H](N)Cc2ccccc2)c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Luo Y, Shoemaker A R, Liu X, et al. Potent and selective inhibitors of Akt kinases slow the progress of tumors in vivo.[J]. Molecular Cancer Therapeutics, 2005, 4[6] 977.