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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $28.05 | Total: $140.25 |
| 1 | 10 | $23.76 | Total: $237.60 |
| 1 | 25 | $20.13 | Total: $503.25 |
| 1 | 50 | $17.16 | Total: $858.00 |
| 1 | 100 | $14.85 | Total: $1,485.00 |
Overview
CCT129202 is an ATP-competitive pan-Aurora inhibitor for Aurora A, Aurora B and Aurora C with IC50 of 0.042 ?M, 0.198 ?M and 0.227 ?M, respectively. It is less potent to FGFR3, GSK3?, PDGFR?, etc.
Chemical Properties
| Molecular Formula | C23H25ClN8OS |
| Molecular Weight | 497.02 |
| CAS Numbers | 942947-93-5 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN(C)c1ccc(cc1)-c1nc2c(N3CCN(CC(=O)Nc4nccs4)CC3)c(Cl)cnc2[nH]1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Chan F, et al. Mol Cancer Ther. 2007, 6[12], 3147-3157.