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GSK1120212
AOB87707
CAS No:871700-17-3
Chemical Name: Trametinib, JTP-74057
492 Items
Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $9.35 | Total: $46.75 |
| 1 | 10 | $7.92 | Total: $79.20 |
| 1 | 25 | $6.71 | Total: $167.75 |
| 1 | 50 | $5.72 | Total: $286.00 |
| 1 | 100 | $4.95 | Total: $495.00 |
Overview
A potent, highly selective and orally active inhibitor of MEK 1 and 2 inhibitor
References:
1: Gilmartin AG, Bleam MR, Groy A, Moss KG, et al., GSK1120212 (JTP-74057) is an inhibitor of MEK activity and activation with favorable pharmacokinetic properties for sustained in vivo pathway inhibition, Clin Cancer Res. 2011 Jan 18. [Epub ahead of print]
Chemical Properties
| Molecular Formula | C26H23FIN5O4 |
| Molecular Weight | 615.39 |
| CAS Numbers | 871700-17-3 |
| Solubility | DMSO |
| Purity | 99% (HPLC) |
Storage and Handling
0°C (short term), -20°C (long term), desiccated