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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $22.10 | Total: $110.50 |
| 1 | 10 | $18.72 | Total: $187.20 |
| 1 | 25 | $15.86 | Total: $396.50 |
| 1 | 50 | $13.52 | Total: $676.00 |
| 1 | 100 | $11.70 | Total: $1,170.00 |
Overview
JSH-150 is a highly selective CDK9 inhibitor with an IC50 of 1 nM.
Chemical Properties
| Molecular Formula | C24H33ClN6O2S |
| Molecular Weight | 505.08 |
| CAS Numbers | 2247481-21-4 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COCCN[C@H]1CC[C@@H](CC1)Nc1cc(-c2csc(NCC3(CCOCC3)C#N)n2)c(Cl)cn1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Beilei Wang, et al. Discovery of 4-[[[4-[5-chloro-2-[[[1s,4s]-4-[[2-methoxyethyl]amino]cyclohexyl]amino]pyridin-4-yl]thiazol-2-yl]amino]methyl]tetrahydro-2H-pyran-4-carbonitrile [JSH-150] as a novel highly selective and potent CDK9 kinase inhibitor. Eur J Med Chem. 13 September 2018.