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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $23.80 | Total: $119.00 |
| 1 | 10 | $20.16 | Total: $201.60 |
| 1 | 25 | $17.08 | Total: $427.00 |
| 1 | 50 | $14.56 | Total: $728.00 |
| 1 | 100 | $12.60 | Total: $1,260.00 |
Overview
JTP-0819958 is a selective linear ubiquitin chain assembly complex (LUBAC) inhibitor with an IC50 of 2.8 ?M[1]. JTP-0819958 suppress LUBAC-mediated NF-kB activation in vitro[2].
Chemical Properties
| Molecular Formula | C17H13NaO4 |
| Molecular Weight | 304.27 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C(O[Na])C1=CC=CC=C1C=CC(C2=C(OC)C=CC=C2)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Ken, Katsuya, Yuji, et al. High-Throughput Screening for Linear Ubiquitin Chain Assembly Complex [LUBAC] Selective Inhibitors Using Homogenous Time-Resolved Fluorescence [HTRF]-Based Assay System.[J]. SLAS discovery advancing life sciences R & D, 2018.