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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $25.50 | Total: $127.50 |
| 1 | 10 | $21.60 | Total: $216.00 |
| 1 | 25 | $18.30 | Total: $457.50 |
| 1 | 50 | $15.60 | Total: $780.00 |
| 1 | 100 | $13.50 | Total: $1,350.00 |
Overview
CAY10462 (CTK8E8405) is an effective and selective inhibitor of the 20-HETE synthase CYP4A11 with an IC50 of 8.8 nM. CAY10462 exhibits nearly 200 times less potent for 1A, 1C, and 3A CYP450 enzymes.
Chemical Properties
| Molecular Formula | C17H27Cl2N3O |
| Molecular Weight | 360.32 |
| CAS Numbers | 502656-68-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN(C)CCCCCCOC(C=C1)=CC=C1N2C=CN=C2.Cl.Cl |
Storage and Handling
0C Short Term, -20C Long Term
References
Nakamura T, et al. Imidazole derivatives as new potent and selective 20-HETE synthase inhibitors. Bioorg Med Chem Lett. 2004 Jan 19;14[2] 333-6.