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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $39.10 | Total: $195.50 |
| 1 | 10 | $33.12 | Total: $331.20 |
| 1 | 25 | $28.06 | Total: $701.50 |
| 1 | 50 | $23.92 | Total: $1,196.00 |
| 1 | 100 | $20.70 | Total: $2,070.00 |
Overview
Desmethyl Erlotinib hydrochloride (OSI 420) is an active metabolite of erlotinib which is an orally active EGFR tyrosin kinase inhibitor with IC50 of 2 and 20 nM for human EGFR and EGFR autophosphorylation in tumor cells.
Chemical Properties
| Molecular Formula | C21H21N3O4 |
| Molecular Weight | 415.87 |
| CAS Numbers | 183320-51-6 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cl.COCCOc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1OCCO |
Storage and Handling
0C Short Term, -20C Long Term
References
Meany HJ, et al. Cancer Chemother Pharmacol. 2008, 62[3], 387-392.