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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $41.65 | Total: $208.25 |
| 1 | 10 | $35.28 | Total: $352.80 |
| 1 | 25 | $29.89 | Total: $747.25 |
| 1 | 50 | $25.48 | Total: $1,274.00 |
| 1 | 100 | $22.05 | Total: $2,205.00 |
Overview
CYP11B2-IN-1 is an effective and selective inhibitor of CYP11B2 with IC50s of 2.3 nM and 142 nM for CYP11B2 and CYP11B1.
Chemical Properties
| Molecular Formula | C18H18FN3O |
| Molecular Weight | 311.35 |
| CAS Numbers | 1356479-78-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | FC=1C=C2N(C(=NC2=CC1)C=3C=C(C(C)(C)O)C=NC3)C4CC4 |
Storage and Handling
0C Short Term, -20C Long Term
References
Hoyt SB, et al. Discovery of Benzimidazole CYP11B2 Inhibitors with in Vivo Activity in Rhesus Monkeys.ACS Med Chem Lett. 2015 Apr 7;6[5] 573-8.