Categories
- PROTAC Linker
- Protein Control Ligand
- Pathway Inhibitors
- Function Modulators
- Activators
- G Protein-Coupled Receptor Ligands
- Nuclear Receptor Ligands
- GDNF Receptors
- TNF Receptors
- Transcription Factors
- Chemokines
- Cytokine Receptors
- Biomarkers and Buffer Solutions
- Molecular Probes
- Stem Cell Research
- Alzheimer's Disease
- Apoptosis
- Cancer Research
- Epigenetics
- Metabolites
- PET/SPECT Imaging Precursors
- Customized Screening Library
- Ultra Pure Pharmacological Standard
- Tissue Microarray (TMA)
- Proteins and Antibodies
- Primary Cells
- ELISA KIT
- Natural Products
- Lab Equipments
- Humanized Mice for PDX Platform
- Rare Chemicals
- Custom Synthesis
- Antibacterial
- Antifungal
- Antioxidant
- Antiviral
- Molecular Glues
- SARS-CoV
Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $130.90 | Total: $654.50 |
| 1 | 10 | $110.88 | Total: $1,108.80 |
| 1 | 25 | $93.94 | Total: $2,348.50 |
| 1 | 50 | $80.08 | Total: $4,004.00 |
| 1 | 100 | $69.30 | Total: $6,930.00 |
Overview
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4 M for the nk-2 receptor in the small intestine of rats.
Chemical Properties
| Molecular Formula | C59H69F3N12O12 |
| Molecular Weight | 1195.25 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC([C@H](NC([C@H](NC([C@@H](NC([C@@H](N)CC(O)=O)=O)CC1=CC=C(O)C=C1)=O)CC2=CNC3=CC=CC=C32)=O)C(N[C@@H](C(N[C@@H](C(N[C@H](C(N)=O)CCCCN)=O)CC4=CNC5=CC=CC=C54)=O)CC6=CNC7=CC=CC=C76)=O)C.OC(C(F)(F)F)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Quartara L, et al. N-terminal truncated analogs of men 10376 as tachykinin NK-2 receptor antagonists. Life Sci. 1992;51[25] 1929-36.