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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $31.45 | Total: $157.25 |
| 1 | 10 | $26.64 | Total: $266.40 |
| 1 | 25 | $22.57 | Total: $564.25 |
| 1 | 50 | $19.24 | Total: $962.00 |
| 1 | 100 | $16.65 | Total: $1,665.00 |
Overview
SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.
Chemical Properties
| Molecular Formula | C25H20N2O3 |
| Molecular Weight | 396.44 |
| CAS Numbers | 174635-53-1 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(N[C@@H](C(OC)=O)C1=CC=CC=C1)(=O)C=2C3=C(N=C(C2)C4=CC=CC=C4)C=CC=C3 |
Storage and Handling
0C Short Term, -20C Long Term
References
Medhurst AD, et, al. In vitro and in vivo characterization of NK3 receptors in the rabbit eye by use of selective non-peptide NK3 receptor antagonists. Br J Pharmacol. 1997 Oct;122[3] 469-76.