[Lys5,MeLeu9,Nle10]-NKA(4-10)

[Lys5,MeLeu9,Nle10]-NKA(4-10)

ATP1883

CAS 137565-28-7

More details

1000 Items

$191.10

$191.10 per mg

Quantity Discount Table - Order More To Get More Price Discount

QuantitymgUnit Price ($/mg or $/Unit)Final Price
15 $124.95 Total: $624.75
110 $105.84 Total: $1,058.40
125 $89.67 Total: $2,241.75
150 $76.44 Total: $3,822.00
1100 $66.15 Total: $6,615.00

Overview

Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).

Chemical Properties

Molecular FormulaC39H65N9O9
Molecular Weight803.99
CAS Numbers137565-28-7
SolubilityDMSO
Purity98% by HPLC
SMILES Code[C@@H](CC1=CC=CC=C1)(NC([C@@H](NC([C@H](CC(O)=O)N)=O)CCCCN)=O)C(N[C@H](C(NCC(N([C@H](C(N[C@@H](CCCC)C(N)=O)=O)CC(C)C)C)=O)=O)C(C)C)=O

Storage and Handling

0C Short Term, -20C Long Term

References

Chassaing et al [1991] Selective agonists of NK-2 binding sites highly active on rat portal vein [NK-3 bioassay]. Neuropeptides 19 91 PMID