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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $118.15 | Total: $590.75 |
| 1 | 10 | $100.08 | Total: $1,000.80 |
| 1 | 25 | $84.79 | Total: $2,119.75 |
| 1 | 50 | $72.28 | Total: $3,614.00 |
| 1 | 100 | $62.55 | Total: $6,255.00 |
Overview
NIK SMI1 is an effective and selective NF-?B inducing kinase (NIK) inhibitor. It also inhibits NIK-catalyzed hydrolysis of ATP to ADP (IC50: 0.23
Chemical Properties
| Molecular Formula | C20H19N3O4 |
| Molecular Weight | 365.38 |
| CAS Numbers | 1660114-31-7 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | COc1cc(nc(c1)-c1cccc(c1)C#C[C@]1(O)CCN(C)C1=O)C(N)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Blaquiere N, et al. Scaffold-Hopping Approach To Discover Potent, Selective, and Efficacious Inhibitors of NF-?B Inducing Kinase. J Med Chem. 2018 Aug 9;61[15] 6801-6813.