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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $45.05 | Total: $225.25 |
| 1 | 10 | $38.16 | Total: $381.60 |
| 1 | 25 | $32.33 | Total: $808.25 |
| 1 | 50 | $27.56 | Total: $1,378.00 |
| 1 | 100 | $23.85 | Total: $2,385.00 |
Overview
APE1-IN-1 is a potent inhibitor of purinepyrimidine endonuclease 1 (APE1) that crosses the blood-brain barrier, exhibits potential antitumor activity, and enhances the cytotoxicity of the alkylating agent [methyl methanesulfonate] on cancer cells.
Chemical Properties
| Molecular Formula | C19H21N3OS2 |
| Molecular Weight | 371.52 |
| CAS Numbers | 524708-03-0 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(C)N1CCc2c(C1)sc(NC(C)=O)c2-c1nc2ccccc2s1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Rai G, et al. Synthesis, biological evaluation, and structure-activity relationships of a novel class of apurinicapyrimidinic endonuclease 1 inhibitors. J Med Chem. 2012 Apr 12;55[7] 3101-12.