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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $76.50 | Total: $382.50 |
| 1 | 10 | $64.80 | Total: $648.00 |
| 1 | 25 | $54.90 | Total: $1,372.50 |
| 1 | 50 | $46.80 | Total: $2,340.00 |
| 1 | 100 | $40.50 | Total: $4,050.00 |
Overview
VU6015929 is an inhibitor of active dual discoidin domain receptor 12 (DDR12)( IC50s of 4.67 nM and 7.39 nM, respectively).
Chemical Properties
| Molecular Formula | C24H19F4N5O2 |
| Molecular Weight | 485.43 |
| CAS Numbers | 2442597-56-8 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | Cn1ccc(n1)-c1cncc(CNc2cc(ccc2F)C(=O)Nc2cccc(OC(F)(F)F)c2)c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Jeffries DE, Borza CM, Blobaum AL,et al.Discovery of VU6015929 A Selective Discoidin Domain Receptor 12 [DDR12] Inhibitor to Explore the Role of DDR1 in Antifibrotic Therapy[1].ACS Med Chem Lett. 2019 Nov 25 ;11[1] 29-33.