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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $147.90 | Total: $739.50 |
| 1 | 10 | $125.28 | Total: $1,252.80 |
| 1 | 25 | $106.14 | Total: $2,653.50 |
| 1 | 50 | $90.48 | Total: $4,524.00 |
| 1 | 100 | $78.30 | Total: $7,830.00 |
Overview
CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the ?-opioid receptor with IC50 of 3.5 nM. It displays over 1200-fold selectivity over ? opioid (IC50=4500 nM) and somatostatin receptors. CTAP(TFA? (103429-32-9 free base) can be used for the study of L-DOPA-induced dyskinesia (LID)
Chemical Properties
| Molecular Formula | C53H70F3N13O13S2 |
| Molecular Weight | 1218.33 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CC(O)C1C(NC(C(NC(C(N)=O)C(O)C)=O)C(C)(C)SSCC(NC(C(N)CC2=CC=CC=C2)=O)C(NC(CC3=CC=C(O)C=C3)C(NC(CC4=CNC5=CC=CC=C54)C(NC(CCCN=C(N)N)C(N1)=O)=O)=O)=O)=O.O=C(O)C(F)(F)F |
Storage and Handling
0C Short Term, -20C Long Term
References
Mitchell J Bartlett, et al. Highly-selective