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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $103.70 | Total: $518.50 |
| 1 | 10 | $87.84 | Total: $878.40 |
| 1 | 25 | $74.42 | Total: $1,860.50 |
| 1 | 50 | $63.44 | Total: $3,172.00 |
| 1 | 100 | $54.90 | Total: $5,490.00 |
Overview
SCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used to study neurological disorders.
Chemical Properties
| Molecular Formula | C28H31NO |
| Molecular Weight | 397.55 |
| CAS Numbers | 322473-89-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | C(N1[C@@]2(C[C@@](O)(C[C@]1(CC2)[H])C3=CC=CC=C3)[H])(C4=C(C)C=CC=C4)C5=C(C)C=CC=C5 |
Storage and Handling
0C Short Term, -20C Long Term
References
Varty GB, et al. The anxiolytic-like effects of the novel, orally active nociceptin opioid receptor agonist 8-[bis[2-methylphenyl]methyl]-3-phenyl-8-azabicyclo[3.2.1]octan-3-ol [SCH 221510]. J Pharmacol Exp Ther. 2008 Aug;326[2] 672-82.