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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $69.70 | Total: $348.50 |
| 1 | 10 | $59.04 | Total: $590.40 |
| 1 | 25 | $50.02 | Total: $1,250.50 |
| 1 | 50 | $42.64 | Total: $2,132.00 |
| 1 | 100 | $36.90 | Total: $3,690.00 |
Overview
BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain barrier permeability and potency, with Kis values of 1.8 nM for MOP and 4.2 nM for NOP.BPR1M97 exhibits anti-injurious effects and antinociceptive effects.
Chemical Properties
| Molecular Formula | C18H18Cl2N2O |
| Molecular Weight | 349.25 |
| CAS Numbers | 2059904-66-2 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | CN1CCc2ccccc2C1CNC(=O)c1ccc(Cl)c(Cl)c1 |
Storage and Handling
0C Short Term, -20C Long Term
References
Chao PK, et al. BPR1M97, a dual mu opioid receptornociceptin-orphanin FQ peptide receptor agonist, producespotent antinociceptive effects with safer properties than morphine. Neuropharmacology. 2019 Jul 3 107678.