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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $253.30 | Total: $1,266.50 |
| 1 | 10 | $214.56 | Total: $2,145.60 |
| 1 | 25 | $181.78 | Total: $4,544.50 |
| 1 | 50 | $154.96 | Total: $7,748.00 |
| 1 | 100 | $134.10 | Total: $13,410.01 |
Overview
6'-GNTI dihydrochloride is a ?-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over recruitment of ?-aspirin 2. 6'-GNTI dihydrochloride only activates the Akt pathway in striatal neurons.
Chemical Properties
| Molecular Formula | C27H29N5O3.2ClH |
| Molecular Weight | 544.47 |
| CAS Numbers | 2410327-94-3 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O[C@]12[C@]34[C@](OC5=C(O)C=CC(C[C@@]2([H])N(CC4)CC6CC6)=C53)([H])C7=C(C8=CC=C(NC(N)=N)C=C8N7)C1.Cl.Cl |
Storage and Handling
0C Short Term, -20C Long Term
References
Schmid CL, et al. Functional selectivity of 6'-guanidinonaltrindole [6'-GNTI] at ?-opioid receptors in striatal neurons. J Biol Chem. 2013;288[31] 22387-22398.