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Quantity Discount Table - Order More To Get More Price Discount
| Quantity | mg | Unit Price ($/mg or $/Unit) | Final Price |
|---|---|---|---|
| 1 | 5 | $73.10 | Total: $365.50 |
| 1 | 10 | $61.92 | Total: $619.20 |
| 1 | 25 | $52.46 | Total: $1,311.50 |
| 1 | 50 | $44.72 | Total: $2,236.00 |
| 1 | 100 | $38.70 | Total: $3,870.00 |
Overview
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the ?-opioid receptor. Dynorphin A (1-10) also blocks NMDA-activated current with an IC50 of 42.0 ?M.
Chemical Properties
| Molecular Formula | C59H95N19O14 |
| Molecular Weight | 1294.53 |
| Solubility | DMSO |
| Purity | 98% by HPLC |
| SMILES Code | O=C([C@H](CCCNC(N)=N)NC([C@H]([C@@H](C)CC)NC([C@H](CCCNC(N)=N)NC([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@@H](NC(CNC(CNC([C@@H](N)CC1=CC=C(O)C=C1)=O)=O)=O)CC2=CC=CC=C2)=O)=O)=O)=O)=O)N3[C@H](C(O)=O)CCC3.CC(O)=O |
Storage and Handling
0C Short Term, -20C Long Term
References
Paterlini G, et al. Molecular simulation of dynorphin A-[1-10] binding to extracellular loop 2 of the kappa-opioidreceptor. A model for receptor activation. J Med Chem. 1997 Sep 26;40[20] 3254-62.